Synthesis of 2-[18F]fluoro-3-[2(S)-2-azetidinylmethoxy]pyridine, a highly potent radioligand for in vivo imaging central nicotinic acetylcholine receptors

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Pharmacology, toxicology, and radiation dosimetry evaluation of [123I]5-I-A-85380, a radioligand for in vivo imaging of cerebral neuronal nicotinic acetylcholine receptors in humans

Drug Development Research ◽

10.1002/ddr.10152 ◽

2003 ◽

Vol 58 (2) ◽

pp. 149-168 ◽

Cited By ~ 11

Author(s):

D. Bruce Vaupel ◽

Srihari R. Tella ◽

David L. Huso ◽

Alexey G. Mukhin ◽

Ira Baum ◽

...

Keyword(s):

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Radiation Dosimetry ◽

Neuronal Nicotinic Acetylcholine Receptors ◽

The Quest for Eldorado: Development of Radioligands for In Vivo Imaging of Nicotinic Acetylcholine Receptors in Human Brain

Current Pharmaceutical Design ◽

10.2174/138161206778559605 ◽

2006 ◽

Vol 12 (30) ◽

Cited By ~ 39

Author(s):

Andrew G. Horti ◽

Victor L. Villemagne

Keyword(s):

Human Brain ◽

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Synthesis and biological evaluation of novel carbon-11 labeled pyridyl ethers: candidate ligands for in vivo imaging of α4β2 nicotinic acetylcholine receptors (α4β2-nAChRs) in the brain with positron emission tomography

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2009.05.021 ◽

2009 ◽

Vol 17 (13) ◽

pp. 4367-4377 ◽

Cited By ~ 6

Author(s):

Yongjun Gao ◽

Hayden T. Ravert ◽

Hiroto Kuwabara ◽

Yingxian Xiao ◽

Christopher J. Endres ◽

...

Keyword(s):

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Biological Evaluation ◽

Emission Tomography ◽

Nicotinic Acetylcholine ◽

Positron Emission ◽

Synthesis And Biological Evaluation ◽

The Brain

In Vivo Imaging of Nicotinic Acetylcholine Receptors in the Central Nervous System

Nicotinic Acetylcholine Receptor Signaling in Neuroprotection ◽

10.1007/978-981-10-8488-1_2 ◽

2018 ◽

pp. 17-44

Author(s):

Masashi Ueda ◽

Yuki Matsuura ◽

Ryosuke Hosoda ◽

Hideo Saji

Keyword(s):

Central Nervous System ◽

Nervous System ◽

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

The Central Nervous System

6-[18F]fluoro-A-85380, a novel radioligand for in vivo imaging of central nicotinic acetylcholine receptors

Life Sciences ◽

10.1016/s0024-3205(00)00635-4 ◽

2000 ◽

Vol 67 (4) ◽

pp. 463-469 ◽

Cited By ~ 35

Author(s):

Andrew G. Horti ◽

Svetlana I. Chefer ◽

Alexey G. Mukhin ◽

Andrei O. Koren ◽

Daniela Gündisch ◽

...

Keyword(s):

In Vivo Imaging ◽

Acetylcholine Receptors ◽

The Prototoxin lynx1 Acts on Nicotinic Acetylcholine Receptors to Balance Neuronal Activity and Survival In Vivo

Neuron ◽

10.1016/j.neuron.2006.07.025 ◽

2006 ◽

Vol 51 (5) ◽

pp. 587-600 ◽

Cited By ~ 89

Author(s):

Julie M. Miwa ◽

Tanya R. Stevens ◽

Sarah L. King ◽

Barbara J. Caldarone ◽

Ines Ibanez-Tallon ◽

...

Keyword(s):

Neuronal Activity ◽

Acetylcholine Receptors ◽

LC-MS Supported Studies on the in Vitro Metabolism of both Enantiomers of Flubatine and the in Vivo Metabolism of (+)-[18F]Flubatine—A Positron Emission Tomography Radioligand for Imaging α4β2 Nicotinic Acetylcholine Receptors

Molecules ◽

10.3390/molecules21091200 ◽

2016 ◽

Vol 21 (9) ◽

pp. 1200 ◽

Cited By ~ 7

Author(s):

Friedrich-Alexander Ludwig ◽

René Smits ◽

Steffen Fischer ◽

Cornelius Donat ◽

Alexander Hoepping ◽

...

Keyword(s):

Positron Emission Tomography ◽

Acetylcholine Receptors ◽

In Vitro Metabolism ◽

Emission Tomography ◽

In Vivo Metabolism ◽

Nicotinic Acetylcholine ◽

Positron Emission

Activation of nicotinic acetylcholine receptors induces long-term potentiation in vivo in the intact mouse dentate gyrus

European Journal of Neuroscience ◽

10.1046/j.1460-9568.2000.00259.x ◽

2000 ◽

Vol 12 (10) ◽

pp. 3741-3747 ◽

Cited By ~ 108

Author(s):

Shogo Matsuyama ◽

Akira Matsumoto ◽

Taira Enomoto ◽

Tomoyuki Nishizaki

Keyword(s):

Dentate Gyrus ◽

Acetylcholine Receptors ◽

Long Term Potentiation ◽

Intact Mouse ◽

Nicotinic Acetylcholine ◽

Term Potentiation

Methanandamide Allosterically Inhibits in Vivo the Function of Peripheral Nicotinic Acetylcholine Receptors Containing the α7-Subunit

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.108.140863 ◽

2008 ◽

Vol 326 (3) ◽

pp. 912-919 ◽

Cited By ~ 14

Author(s):

Urszula Baranowska ◽

Manfred Göthert ◽

Radosław Rudź ◽

Barbara Malinowska

Keyword(s):

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

Α7 Subunit

In vivo quantification of the greater densities of alpha4beta2* nicotinic acetylcholine receptors in smokers compared to non-smokers

NeuroImage ◽

10.1016/j.neuroimage.2006.04.136 ◽

2006 ◽

Vol 31 ◽

pp. T153 ◽

Cited By ~ 2

Author(s):

Alane S. Kimes ◽

S. Chefer ◽

C.S. Contoreggi ◽

A. Hall ◽

A. Horti ◽

...

Keyword(s):

Acetylcholine Receptors ◽